Palonosetron hydrochloride ( Aloxi; RS 25259-197 )

产品货号. M11463 CAS No. 135729-62-3

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产品名称

Palonosetron hydrochloride
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

Palonosetron (INN, trade name Aloxi) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting (CINV).
产品描述

Palonosetron (INN, trade name Aloxi) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting (CINV). It is the most effective of the 5-HT3 antagonists in controlling delayed CINV nausea and vomiting that appear more than 24 hours after the first dose of a course of chemotherapy and is the only drug of its class approved for this use by the U.S. Food and Drug Administration. As of 2008, it is the most recent 5-HT3 antagonist to enter clinical use.
同义词

Aloxi; RS 25259-197
通路

Endocrinology/Hormones
靶点

5-HT Receptor
受体

5-HT
研究领域

Cardiovascular Disease
适应症

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1.Grunberg SM, Koeller JM. Expert Opin PharmacOthers. 2003 Dec;4(12):2297-303.

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